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Toplam kayıt 6, listelenen: 1-6
Synthesis and Carbonic Anhydrase Inhibitory Effects of Novel Sulfamides Derived from 1-Aminoindanes and Anilines
(Wiley-V C H Verlag Gmbh, 2014)
Three 1-aminoindanes, four anilines and BnOH or t-BuOH were reacted with chlorosulfonyl isocyanate to give sulfamoyl carbamates. Pd-C catalysed hydrogenolysis reactions of carbamates or deprotection of the Boc group of the ...
In vitro inhibition of alpha-carbonic anhydrase isozymes by some phenolic compounds
(Pergamon-Elsevier Science Ltd, 2011)
Carbonic anhydrase inhibitors (CAIs) are a class of pharmaceuticals used as antiglaucoma agents, diuretics, antiepileptics, in the management of mountain sickness, gastric and duodenal ulcers, neurological disorders or ...
9,10-Dibromo-N-aryl-9,10-dihydro-9,10-[3,4]epipyrroloanthracene-12,14-diones: Synthesis and Investigation of Their Effects on Carbonic Anhydrase Isozymes I, II, IX, and XII
(Wiley-V C H Verlag Gmbh, 2016)
N-substituted maleimides were synthesized from maleic anhydride and primary amines. 1,4-Dibromodibenzo[e,h]bicyclo-[2,2,2]octane-2,3-dicarboximide derivatives (4a-f) were prepared by the [4+2] cycloaddition reaction of ...
Synthesis and Determination of Some Biological Activities of Novel 2,4-Dinitrophenyl Derivatives
(Wiley-V C H Verlag Gmbh, 2015)
The antioxidant and radical scavenging activities of the synthesized compounds 3, 5, and 6 were determined by various in vitro assays such as 2,2-azino-bis(3-ethylbenzthiazoline-6-sulfonic acid radical (ABTS(+)) scavenging, ...
Novel eugenol derivatives: Potent acetylcholinesterase and carbonic anhydrase inhibitors
(Elsevier Science Bv, 2017)
Eugenol was used as starting material to obtain some phenolic compounds. The synthesis of these phenolic compounds was performed in a two-step procedure. The structures of the formed products (novel eugenol derivatives ...
N-Acylsulfonamides strongly inhibit human carbonic anhydrase isoenzymes I and II
(Pergamon-Elsevier Science Ltd, 2015)
Sulfonamides represent a significant class of biologically active compounds that inhibit carbonic anhydrase (CA, EC.: 4.2.1.1) isoenzymes involved in different pathological and physiological events. Sulfonamide CA inhibitors ...