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Toplam kayıt 8, listelenen: 1-8
Synthesis and Carbonic Anhydrase Inhibitory Effects of Novel Sulfamides Derived from 1-Aminoindanes and Anilines
(Wiley-V C H Verlag Gmbh, 2014)
Three 1-aminoindanes, four anilines and BnOH or t-BuOH were reacted with chlorosulfonyl isocyanate to give sulfamoyl carbamates. Pd-C catalysed hydrogenolysis reactions of carbamates or deprotection of the Boc group of the ...
In vitro inhibition of alpha-carbonic anhydrase isozymes by some phenolic compounds
(Pergamon-Elsevier Science Ltd, 2011)
Carbonic anhydrase inhibitors (CAIs) are a class of pharmaceuticals used as antiglaucoma agents, diuretics, antiepileptics, in the management of mountain sickness, gastric and duodenal ulcers, neurological disorders or ...
9,10-Dibromo-N-aryl-9,10-dihydro-9,10-[3,4]epipyrroloanthracene-12,14-diones: Synthesis and Investigation of Their Effects on Carbonic Anhydrase Isozymes I, II, IX, and XII
(Wiley-V C H Verlag Gmbh, 2016)
N-substituted maleimides were synthesized from maleic anhydride and primary amines. 1,4-Dibromodibenzo[e,h]bicyclo-[2,2,2]octane-2,3-dicarboximide derivatives (4a-f) were prepared by the [4+2] cycloaddition reaction of ...
Carbonic anhydrase I and II autoantibodies in Behcet's disease
(Publisaude-Edicoes Medicas Lda, 2017)
Background: Behcet's disease ( BD) is a vasculitis, seen more frequently around the Mediterranean and the Far East, and evinces with oral and genital ulcerations, skin lesions and uveitis. Carbonic anhydrase ( CA) is a ...
Inhibition Profiles of Some Symmetric Sulfamides Derived from Phenethylamines on Human Carbonic Anhydrase I, and II Isoenzymes
(Wiley-V C H Verlag Gmbh, 2021)
In this work, the inhibitory effect of some symmetric sulfamides derived from phenethylamines were determined against human carbonic anhydrase (hCA) I, and II isoenzymes, and compared with standard compound acetazolamide. ...
Synthesis and Determination of Some Biological Activities of Novel 2,4-Dinitrophenyl Derivatives
(Wiley-V C H Verlag Gmbh, 2015)
The antioxidant and radical scavenging activities of the synthesized compounds 3, 5, and 6 were determined by various in vitro assays such as 2,2-azino-bis(3-ethylbenzthiazoline-6-sulfonic acid radical (ABTS(+)) scavenging, ...
Novel eugenol derivatives: Potent acetylcholinesterase and carbonic anhydrase inhibitors
(Elsevier Science Bv, 2017)
Eugenol was used as starting material to obtain some phenolic compounds. The synthesis of these phenolic compounds was performed in a two-step procedure. The structures of the formed products (novel eugenol derivatives ...
N-Acylsulfonamides strongly inhibit human carbonic anhydrase isoenzymes I and II
(Pergamon-Elsevier Science Ltd, 2015)
Sulfonamides represent a significant class of biologically active compounds that inhibit carbonic anhydrase (CA, EC.: 4.2.1.1) isoenzymes involved in different pathological and physiological events. Sulfonamide CA inhibitors ...