Ara
Toplam kayıt 3, listelenen: 1-3
Rosmarinic acid: a potent carbonic anhydrase isoenzymes inhibitor
(2014-08-15)
Rosmarinic acid is a water-soluble ester of ca eic acid and 3,4-dihydroxyphenyllactic acids, and is mainly found in plant species including Boraginaceae and Lamiaceae. In this research, we determined the inhibition property ...
Novel Sulphamides and Sulphonamides Incorporating the Tetralin Scaffold as Carbonic Anhydrase and Acetylcholine Esterase Inhibitors
(2013-09-17)
Reactions of amino, aminomethyl tetralins and benzyl alcohol with chlorosulphonyl isocyanate (CSI)
afforded sulphamoyl carbamates. The sulphamoyl carbamates were converted to sulphamides by
palladium-catalysed hydrogenolysis. ...
(3,4-Dihydroxyphenyl)(2,3,4-trihydroxyphenyl)methanone and its derivatives as carbonic anhydrase isoenzymes inhibitors
(Journal of Enzyme Inhibition and Medicinal Chemistry, 2013-04)
In this study, we have synthesised (3,4-dihydroxyphenyl)(2,3,4-trihydroxyphenyl)methanone and a series of its
derivatives (5, 13–16) and tested the ability of these compounds to inhibit two metalloenzyme human carbonic ...